Factory 99% Flupirtine Maleate Powder CAS 75507-68-5 Relieve Pain Flupirtine Maleate

• Customization: Available
• Powder: Yes
• Customized: Customized
• Model NO.: A69
• Certification: GMP, HSE, ISO 9001, USP, BP
• Suitable for: Adult
• State: Powder
• Purity: >99%
• Name: Flupirtine Maleate
• Appearance: White Powder
• Assay: 99%
• CAS: 75507-68-5
• OEM: Available
• Sample: Available
• Suitable: Adult
• Function: Relieve Pain
• MOQ: 10g
• Transport Package: Foil Bag
• Specification: 99
• Trademark: /
• Origin: China
• Production Capacity: 10000 Kgs Per Month

Product Description

Product Name	Flupirtine Maleate
Appearance	White Powder
CAS NO.	75507-68-5
Molecular Formula	C19H21FN4O6
Storage	Keep in a cool, dry, dark location

 

Flupirtine maleate is a selective neuronal potassium channel openers, readily absorbed orally with analgesic, muscle relaxation and neuroprotective three efficacy, pain showed analgesic effects to a variety of causes.  As in the hot plate test, intensity of flupirtine (ED50 32mg/Kg, Ig) is about half of the 2 times of  paracetamol 10 times stronger. In the pulp electrical stimulation test of conscious dogs, the intensity of pain (ED50, 3.5mg/Kg, intragastric administration) was comparable to that of Zosin.

 

1. Analgesic Therapy: It is primarily used for the symptomatic treatment of pain, particularly in conditions where non-opioid analgesics are preferred or required.
2. Musculoskeletal Disorders: Commonly prescribed for alleviating pain associated with muscle and skeletal conditions such as acute and chronic back pain, neck pain, and joint pain.
3. Postoperative Pain Management: Employed in the management of moderate to severe pain following surgical procedures, especially where opioid use is to be minimized.

1. Non-Opioid Analgesic Action: Flupirtine exerts its analgesic effect through a unique mechanism that does not involve opioid receptors, reducing the risk of addiction, tolerance, and certain side effects associated with opioids.
2. Central Nervous System Modulation: It modulates neurotransmitter systems in the central nervous system, particularly by inhibiting the release of excitatory neurotransmitters and enhancing inhibitory pathways, leading to pain relief.
3. Anti-Inflammatory Effect (Indirect): Although not a classical anti-inflammatory drug, flupirtine may indirectly reduce inflammation-related pain by modulating the pain perception process, contributing to an overall improvement in pain symptoms.